Synthesis, structure–activity relationships and stereochemical investigations of new tricyclic pyridazinone derivatives as potential STAT3 inhibitors
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منابع مشابه
Novel Tricyclic Cyanopyrrolidine Derivatives as Dpp4 Inhibitors: an Improved Synthesis of Tricyclic Α-cycnopyrrolidine from Camphor
An improved multistep synthesis of tricyclic α-cyanopyrrolidine from camphor is presented. The synthesis was carried out by maintaining the cyano group in the form of an amide and its regeneration after the completion of the necessary chemical transformation of a particular functional group. The tricyclic α-cyanopyrrolidine prepared was used to synthesize two novel compounds of DPP4 (Dipeptidyl...
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ژورنال
عنوان ژورنال: MedChemComm
سال: 2013
ISSN: 2040-2503,2040-2511
DOI: 10.1039/c3md00095h